Synthesis of heteroaryl substituted α-mercapto acids from thiomalic acid using hexafluoroacetone as protecting and activating reagent

Ksenia Pumpor; Elisabeth Windeisen; Klaus Burger

doi:10.1002/jhet.5570400306

Synthesis of heteroaryl substituted α-mercapto acids from thiomalic acid using hexafluoroacetone as protecting and activating reagent

Ksenia Pumpor, Elisabeth Windeisen, Klaus Burger^*

^*Corresponding author for this work

Institute of Biochemistry

University of Leipzig

16 Citations (Scopus)

Abstract

The synthesis of heterocyclic α-mercapto acids starting from (RS)-thiomalic acid using hexafluoroacetone as protecting and activating agent is described. The new compounds are useful building blocks for peptide and depsipeptide modification as well as for drug design.

Original language	English
Journal	Journal of Heterocyclic Chemistry
Volume	40
Issue number	3
Pages (from-to)	435-442
Number of pages	8
ISSN	0022-152X
DOIs	https://doi.org/10.1002/jhet.5570400306
Publication status	Published - 2003

Research Areas and Centers

Academic Focus: Center for Infection and Inflammation Research (ZIEL)

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This output contributes to the following UN Sustainable Development Goals (SDGs)

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10.1002/jhet.5570400306

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title = "Synthesis of heteroaryl substituted α-mercapto acids from thiomalic acid using hexafluoroacetone as protecting and activating reagent",

abstract = "The synthesis of heterocyclic α-mercapto acids starting from (RS)-thiomalic acid using hexafluoroacetone as protecting and activating agent is described. The new compounds are useful building blocks for peptide and depsipeptide modification as well as for drug design.",

author = "Ksenia Pumpor and Elisabeth Windeisen and Klaus Burger",

year = "2003",

doi = "10.1002/jhet.5570400306",

language = "English",

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pages = "435--442",

journal = "Journal of Heterocyclic Chemistry",

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T1 - Synthesis of heteroaryl substituted α-mercapto acids from thiomalic acid using hexafluoroacetone as protecting and activating reagent

AU - Pumpor, Ksenia

AU - Windeisen, Elisabeth

AU - Burger, Klaus

PY - 2003

Y1 - 2003

N2 - The synthesis of heterocyclic α-mercapto acids starting from (RS)-thiomalic acid using hexafluoroacetone as protecting and activating agent is described. The new compounds are useful building blocks for peptide and depsipeptide modification as well as for drug design.

AB - The synthesis of heterocyclic α-mercapto acids starting from (RS)-thiomalic acid using hexafluoroacetone as protecting and activating agent is described. The new compounds are useful building blocks for peptide and depsipeptide modification as well as for drug design.

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U2 - 10.1002/jhet.5570400306

DO - 10.1002/jhet.5570400306

M3 - Journal articles

AN - SCOPUS:0037961038

SN - 0022-152X

VL - 40

SP - 435

EP - 442

JO - Journal of Heterocyclic Chemistry

JF - Journal of Heterocyclic Chemistry

IS - 3

ER -

Synthesis of heteroaryl substituted α-mercapto acids from thiomalic acid using hexafluoroacetone as protecting and activating reagent

Abstract

Research Areas and Centers

UN SDGs

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