α-fluoromethyl tryptophans via imino ene reaction

S. N. Osipov; N. M. Kobel'Kova; A. F. Kolomiets; K. Pumpor; B. Koksch; K. Burger

doi:10.1055/s-2001-16054

α-fluoromethyl tryptophans via imino ene reaction

S. N. Osipov, N. M. Kobel'Kova, A. F. Kolomiets, K. Pumpor, B. Koksch, K. Burger^*

^*Korrespondierende/r Autor/-in für diese Arbeit

Institut für Biochemie

Universität Leipzig

14 Zitate (Scopus)

Abstract

A preparative simple synthesis of α-fluoromethyl tryptophans is described. The new method is based on a non-catalytic imine ene reaction of highly electrophilic imines derived from methyl bromodifluoro- and trifluoropyruvate, and 1-sulfonyl-3-methylene indolines.

Originalsprache	Englisch
Zeitschrift	Synlett
Ausgabenummer	8
Seiten (von - bis)	1287-1289
Seitenumfang	3
ISSN	0936-5214
DOIs	https://doi.org/10.1055/s-2001-16054
Publikationsstatus	Veröffentlicht - 2001

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Forschungsschwerpunkt: Infektion und Entzündung - Zentrum für Infektions- und Entzündungsforschung Lübeck (ZIEL)

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10.1055/s-2001-16054

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title = "α-fluoromethyl tryptophans via imino ene reaction",

abstract = "A preparative simple synthesis of α-fluoromethyl tryptophans is described. The new method is based on a non-catalytic imine ene reaction of highly electrophilic imines derived from methyl bromodifluoro- and trifluoropyruvate, and 1-sulfonyl-3-methylene indolines.",

author = "Osipov, \{S. N.\} and Kobel'Kova, \{N. M.\} and Kolomiets, \{A. F.\} and K. Pumpor and B. Koksch and K. Burger",

year = "2001",

doi = "10.1055/s-2001-16054",

language = "English",

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journal = "Synlett",

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AU - Osipov, S. N.

AU - Kobel'Kova, N. M.

AU - Kolomiets, A. F.

AU - Pumpor, K.

AU - Koksch, B.

AU - Burger, K.

PY - 2001

Y1 - 2001

N2 - A preparative simple synthesis of α-fluoromethyl tryptophans is described. The new method is based on a non-catalytic imine ene reaction of highly electrophilic imines derived from methyl bromodifluoro- and trifluoropyruvate, and 1-sulfonyl-3-methylene indolines.

AB - A preparative simple synthesis of α-fluoromethyl tryptophans is described. The new method is based on a non-catalytic imine ene reaction of highly electrophilic imines derived from methyl bromodifluoro- and trifluoropyruvate, and 1-sulfonyl-3-methylene indolines.

UR - https://www.scopus.com/pages/publications/0034902611

U2 - 10.1055/s-2001-16054

DO - 10.1055/s-2001-16054

M3 - Journal articles

AN - SCOPUS:0034902611

SN - 0936-5214

SP - 1287

EP - 1289

JO - Synlett

JF - Synlett

IS - 8

ER -

α-fluoromethyl tryptophans via imino ene reaction

Abstract

UN SDGs

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